Kiwon lafiyaShirye-shirye

Da miyagun ƙwayoyi "Hydroxyzine": umarnin don amfani, analogs da kuma sake dubawa

Diphenylmethane Kalam na abu ne a wajen "Hydroxyzine". User aikace-aikace ya furta cewa, abu ne mai farin lafiya foda, mai narkewa a cikin ruwa da kuma odorless. 374,9 grams da mole ne kwayoyin nauyi na fili.

Clinico-pharmacological kungiyar

Da miyagun ƙwayoyi yana da magani mai kantad da hankali, anxiolytic sakamako. Wannan bayani ne game da hana ruwa guda sakamako a kan ayyuka na wasu subcortical Tsarin na tsakiya m tsarin, kazalika da tarewa mataki a kan tsakiyar H_1-histamine da m-cholinergic rabe.

"Hydroxyzine" miyagun ƙwayoyi analogues da furta kwantad da hankali da kuma m anxiolytic aiki. Da haramta motsa sakamako a kan fahimi damar iya yin komai, inganta da hankali da kuma ƙwaƙwalwar. Qwaqwalwa ne qwarai dogara da buri ba ya faruwa bayan shafe tsawon amfani da ciwo ba a lura. Har ila yau bayyana anticholinergic, antihistamine, antispasmodic mataki. "Hydroxyzine" sauqaqa spasms of m tsoka, sa'an nan haddasa bronchodilatory da analgesic effects, ya mallaka antiemetic mataki da kuma matsakaiciya hana ruwa guda sakamako a kan na ciki mugunya. . Amya, dermatitis, eczema, itching, da dai sauransu rage-rage a lokacin far nufin "Atarax" (hydroxyzine - aiki abu).
Guide ya furta cewa, kwantad da hankali shi ne cimma, yawanci a cikin 10 to 45 minutes bayan ingestion (dangane da tsari da miyagun ƙwayoyi), anti-histamine - sa'a daya bayan ingestion. A marasa lafiya fama da cutar hanta, wani antihistaminic sakamako za a iya sa ran a cikin 96 hours.

Ba alama mutagenic da carcinogenic mataki da miyagun ƙwayoyi.

Pharmacokinetics

Lokacin da ingested da miyagun ƙwayoyi ne hanzari tunawa daga cikin gastrointestinal fili, C_max akwai a sa'o'i biyu. Shiri "Hydroxyzine" ratsa cikin mahaifa da kuma jini-kwakwalwa shamaki (mataki na maida hankali a fetal kyallen takarda mafi girma daga cikin masu juna biyu kyallen takarda). A kan aiwatar da hanta metabolism kafa cetirizine - manyan metabolite. Darajar T_1 / 2 ko da kuwa yana da shekaru na haƙuri kuma zai iya zama 7 hours ga yara shekaru 2-10 shekaru, 20 hours ga manya, 29 hours ga tsofaffi da kuma tsofaffi. a marasa lafiya tare da cutar hanta iya karu zuwa 37 hours. Kawar ne da za'ayi ga mafi part da kodan (0.8% a cikin ainihin form).

alamomi

"Hydroxyzine Hydrochloride" da ake amfani da su:

  • kashe tashin hankali da kuma hyperexcitability na juyayi tsarin.
  • a lokacin janyewar a mutane fama da giya dogara.
  • warkewa magani daga psychoneurotic cuta.
  • kamar yadda wani ɓangare na m magani a cikin postoperative zamani da kuma bayan wasu sun ji rauni.
  • premedication.
  • don rage ciki danniya, kowa yana da tashin hankali, daidaituwa dawo da matakai, a lura da tsari cututtuka.
  • ya kawar da cututtuka na eczema, itchy dermatosis, urticaria, atopic dermatitis.
  • domin antiemetic mataki nuna.

Contraindications da miyagun ƙwayoyi "Hydroxyzine Canon"

Reviews na likitoci nuna cewa da miyagun ƙwayoyi ba da shawarar a sami:

  • marasa lafiya fama da glaucoma.
  • prostate hypertrophy (prostate).
  • marasa lafiya a wanda bãbu ya karu kãmun aiki;
  • marasa lafiya da myasthenia gravis.
  • marasa lafiya da suke yi jinya na koda da hanta gazawar;
  • marasa lafiya da gigin-tsufa.

Da miyagun ƙwayoyi ne contraindicated a cikin:

  • mata masu juna biyu.
  • marasa lafiya da porphyria.
  • nono lokacin (lokacin da magani ya kamata bari nono madarar uwarsa).
  • rashin lafiyan bayyananen for constituting sashi (as a kuma waɗannan lokuta inda a baya alama hypersensitivity zuwa wasu wanda aka samu cetirizine, aminophylline, piperazine ko ethylene diamine).
  • a lokacin aiki da kuma bayarwa.

Game da illa

Marasa lafiya za su wahala daga sleepiness, tasbĩhi janar wani rauni, dizziness da kuma ciwon kai, a farkon miyagun ƙwayoyi far "Hydroxyzine". Reviews da marasa lafiya bi da tare da wannan wakili, ce da wadannan illa:

  • rashin lafiyan halayen, palpitations, tashin zuciya.
  • urinary riƙewa, da kuma maƙarƙashiya.
  • rashin ruwa da ake iya gani mucous membranes, ta ƙara sweating.
  • Heart hangen nesa (yiwu a take hakkin masauki).
  • ragewan jini, ta ƙara hanta enzyme aiki;
  • iya samun bronchospasm.

Very rare bayyanuwar seizures, tsãwa da disorientation, ataxia, paradoxical ruri, kuma Ya ƙãra motor aiki a cikin yin amfani da kayan aikin.

yawan abin sama

Fifiko kira gag reflex ko da ciki an wanke da wani yawan abin sama da miyagun ƙwayoyi "Hydroxyzine". Umurnai na amfani sanar da cewa a wasu lokuta ya zama dole idanu haƙuri da harshen damo, da gabatarwar sodium benzoate, maganin kafeyin, norepinephrine, kuma ko da jini musanya, suna da za'ayi duk matakan da suka dace domin tabbatar da dace aiki na jiki. Specific antidotes da kayan aiki na da, hemodialysis ba za shi barata.

Mafi sau da yawa, wadannan effects ne reversible ko su bayyanar cututtuka bace bayan wani kullum sashi na bita.

sashi

Da miyagun ƙwayoyi ne gudanar da baki ko da intramuscular allura. A kashi dogara nosologies, shekaru na haƙuri kuma siffar a cikin abin da miyagun ƙwayoyi da aka saki "Hydroxyzine".

Umarnin don amfani da shawara cewa symptomatic magani ga tashin hankali ciwo, adult shawarar ci na 25 zuwa 100 MG na bijiro da batun kafa abu a lokacin da rana. Da aka fi amfani sashi na 12.5 MG da safe da kuma a abincin rana da kuma 25 - da yamma.
A cikin shimfiɗar jariri, preoperatively amfani zuwa 1 MG da kg na jiki nauyi da yamma rana kafin da kuma 60 minutes kafin hanya.

Domin manufar premedication aka gudanar a manya "Hydroxyzine" a wani kashi na 50-200 MG na miyagun ƙwayoyi da baki ko a cikin nau'i na intramuscular injections na 1.5-2.5 MG da kg na haƙuri nauyi gudanar sa'a daya kafin tiyata.

Domin manufar taimako na itching tasiri sashi ne daga 25 zuwa 100 MG a 3-4 raba allurai.

Yara daga shekara guda zuwa shekaru 6 da kashi bai wuce 1-2.5 MG da kg na jiki nauyi per day a raba allurai.

A wannan dosing regimen yara a ƙarƙashin da shekaru 6 da shekaru da aka sanya wa 1-2 MG da kg na jiki nauyi a lokacin da rana.

Matsakaicin kullum kashi dauke su 300 MG. Matsakaicin guda kashi - 200 MG.

Tsofaffi qaddamarwa na far bada shawarar a rabin sashi.

Hanta da koda gazawar bukatar gyara daga cikin sashi daga cikin miyagun ƙwayoyi "Hydroxyzine".

Guide yayi kashedin cewa a cimma iyakar warkewa sakamako m bayani ne gudanar intramuscularly, zurfin 50-100 MG da guda kashi. Yana da shawarar Drug Administration dabaru domin 4-6 hours.

A halin tababbu, da magani ne amfani a wani sashi na 300 MG ga kwana. A tsawon lokaci da wannan magani ne 4 makonni.

A hali na bayyanuwar illa kamar wani rauni, drowsiness, ba ya hana a cikin 'yan kwanaki, da kashi ya kamata a rage.

rigakafi

Duk da yake gabatarwar "Hydroxyzine" daga "adrenaline" šauki kasa tasiri.

Da miyagun ƙwayoyi yana da wani reinforcing sakamako a kan magani mai kantad da hankali sakamako na narcotic analgesics jerin, giya, tranquilizers, barbiturates, kwayoyi amfani da nufin hypnotic da sauran kwayoyi da depress CNS aiki.

Ba da shawarar hadin gwiwa aikace-aikace na abu ko holinoblokatorami da Mao hanawa.

Lokacin hade tare da hanyar shan phenytoin anticonvulsant sakamako rage-rage daga liyafar na karshen.

Makaruhai lokaci daya aikace-aikace na miyagun ƙwayoyi da cholinesterase blockers.

A sakamakon kara jini taro na miyagun ƙwayoyi iya bauta wa da aikace-aikace da hanawa na hanta enzymes.

Lokaci daya da magani tare da jamiái wanda hana aiki na CNS, ko da holinoblokatorami bukatar sashi gyara.

Tare da babban kula dole ne a wajabta wa marasa lafiya da ciwon propensity ga fibrillation ko da ake ji antiarrhythmics, kazalika a cikin wadanda marasa lafiya da suke predisposed zuwa convulsive manifestations. A far ne a contraindication ga yin amfani da giya. Idan dole, hali gwaje-gwaje a kan allergies liyafar "Hydroxyzine" to soke har zuwa kwanaki 5 kafin Jirgi jarrabawa. Tsanaki ake bukata sa'ad da yin amfani da miyagun ƙwayoyi da kuma wani abin hawa iko lokaci direbobi da kuma marasa lafiya, da fasahohin da bukatar babban taro.

Ya kamata a haifa tuna cewa amfani da injectables ne kawai zai yiwu ta intramuscular allura. Subcutaneous allura na abin hawa ko shigar azzakari cikin farji na karshen a manyan tasoshin zai iya sa nama lalacewa.

Far da wannan kayan aiki na iya vyzyvavt ƙarya sakamakon prick gwajin.

Sharuddan da yanayi na yin amfani da ajiya

Wajibi ne a cikin wajabta kasancewar wani sayen magani ga miyagun ƙwayoyi "Hydroxyzine".

Umurnai na amfani ya ce na baka siffofin da miyagun ƙwayoyi ba adana fiye da shekaru 5.

"Hydroxyzine". shedu

A yara, da yin amfani da kudi a karkashin Hyperactivity, rage hankali span taimaka da yaro ya zama m, mayar da hankali da kuma m, gusar da yanayi swings. A daidai wannan lokaci da magani daga miyagun ƙwayoyi "Atarax" ( "Hydroxyzine") umarnin don amfani da tabbatar da cewa aiki da lamarinsa na yaro zama guda. Side effects ne rare.

Bisa ga maganganun da marasa lafiya, da ake ji a wasu lokuta "Hydroxyzine" (analogues da miyagun ƙwayoyi), shi ya bi da cewa shi a kwantar da hankula da kuma yarda da kai zuwa mafi girma har fiye da wasu kwayoyi. Tsoro harin da rashin barci da abu inganta mafi barci da kuma sauti barci. Duk da haka, kau da miyagun ƙwayoyi da farko 'yan kwanaki na wani nauyi kuɗin fito a cikin tsari na fadowa barci, amma, bisa manufa, da sakamako daga far ne sosai arfafa.

A farashin da miyagun ƙwayoyi

Saya da miyagun ƙwayoyi "Hydroxyzine" takwarorinsu, a matsayin wani ɓangare na abin da ya ƙunshi hydroxyzine, na iya zama wani kantin magani a kan takardar sayen magani. Price ne 270-300 rubles da 25 Allunan na 25 MG.

"Hydroxyzine". Kamancin

Kamancin na "Hydroxyzine" ne: "Hydroxyzine Canon", "Atarax", "Masmoram", "Ateraks", "Hydroxyzine", "Hydroxyzine Hydrochloride", "Alamon", "Duraks".

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