Kiwon lafiyaShirye-shirye

"Metoprolol": reviews, alamomi don amfani, wa'azi da analogues

Me ya sa zan bukaci magani "Metoprolol"? Shedu da wannan shiri, ta saki siffofin, abun da ke ciki, da kuma illa aka gabatar a kasa. Mu kuma gaya muku game da abin da yake Contra-alamomi da miyagun ƙwayoyi, a cikin abin da kashi ya kamata a dauka idan akwai sauran analogues.

A abun da ke ciki na miyagun ƙwayoyi da ta saki siffofin

A abin da fom da aka sayar da magani "Metoprolol"? Shedu ce cewa kantin magani za a iya samu iri uku da miyagun ƙwayoyi. Ka yi la'akari da batun na cikin tsari da kuma tsarin a more daki-daki.

  • Allunan. Yana dauke da aiki bangaren kamar metoprolol tartrate (100, 50 da kuma 25 milligrams). Bugu da kari, da medicament qunshi karin aka gyara da kuma wani colloidal silica anhydrous, microcrystalline cellulose, sodium carboxymethylstarch (irin A) da kuma magnesium stearate. A sayar da medicament samu 50, 10, 30, 20 ko 40 Allunan da fakitin.
  • Allunan da ci saki Properties ( "metoprolol succinate") mai rufi Allunan. Sun dauke da irin wannan aiki abubuwa da kuma excipients. A Pharmacy irin magani za a iya samu ta hanyar 30, 20 ko 10 Allunan da fakitin.
  • Da mafita ga igiyar jini injections a ampoules na 5 ml. A sayar da miyagun ƙwayoyi zo a cikin wani kartani kwalin 10 vials.

A pharmacological kaddarorin da miyagun ƙwayoyi

Abin da ake nufi magani "Metoprolol"? Alamomi ga yin amfani da kayan aiki za a gabatar a kasa. Yanzu ina so in gaya maka game da abin da yana da pharmacological Properties daga cikin miyagun ƙwayoyi.

Ya ce magani nasa ne a cardioselective beta-adrenergic blockers. Ba ya nuna membrane tabbatar da dorewar Properties kuma yana da wani ciki sympathomimetic aiki. Duk da haka, da aiki da miyagun ƙwayoyi ne an antihypertensive, antiarrhythmic da antianginal wakili.

A medicament ne iya rage mita na haƙuri da zuciya rate, rage tsokar contractility da excitability, m AV-madugu da kuma rage tsokar oxygen bukatar.

Matsayin mai mulkin, da antihypertensive sakamako da aka lura a marasa lafiya ne kawai bayan kwana goma sha huɗu bayan da shan miyagun ƙwayoyi. A medicament rage mita na kai hare-hare tare da supraventricular tachycardia, angina pectoris da atrial fibrillation. A sakamakon haka, al'ada zuciya kari na haƙuri.

Allunan tare da jinkiri saki ( "metoprolol succinate") da wani gagarumin amfani a kan al'ada. Su ka damar kula da akai taro na aiki kashi a cikin jini, sa'an nan samar da mai kyau warkewa sakamako a ko'ina cikin yini. Ya kamata kuma a lura da cewa mataki na "Metoprolol succinate" taimaka wajen rage hadarin bradycardia da wani rauni, to a karami har, rinjayar da m tsokoki na bronchi.

Pharmacokinetics (sha, metabolism da kuma tukar tumbi da miyagun ƙwayoyi)

Game da alamomi don amfani lekarstvai data kasance "Metoprolol" miyagun ƙwayoyi analogues bayyana a kasa, amma yanzu bari mu magana game da pharmacokinetic halaye.

Wannan yana nufin sosai da sauri kuma kusan gaba daya (game da 95%) ne tunawa. Matsakaicin jini taro mafi yawa ana kai bayan 50-110 minti bayan ingestion.

A farko aikace-aikace na miyagun ƙwayoyi bioavailability ne 50%. Maimaita ta ƙãra zuwa 70%. Af, da amfani da abinci mai qara bioavailability na miyagun ƙwayoyi da 20-40%. shi kuma qara idan haƙuri yana da hanta cirrhosis. Sadarwa tare da sunadarai a kan talakawan 10%.

Ya ce medicament da ke shiga cikin placental da jini-kwakwalwa shinge. Har ila yau, a kananan yawa, shi tsaye a waje da kuma cikin nono.

Da miyagun ƙwayoyi ne metabolized a cikin hanta. Kuma metabolites da pharmacological aiki. Game da 5% na Agent excreted da kodan canzawa. Haƙuri Far tare da rage koda aiki na bukatar rage ko wasu gyara kashi. Duk da haka, disturbances a hanta aiki na iya rage gudu metabolism na kwayoyi. A wannan yanayin, da sashi ya kamata a rage.

Magani "Metoprolol": alamomi ga yin amfani da

Akwai quite babban jerin pathological yanayi a wanda da miyagun ƙwayoyi ne gudanar. Bari mu auna su.

  • akathisia, wanda aka sa ta antipsychotics.
  • jijiya hauhawar jini na 1st da 2nd digiri na jijiya hauhawar jini (watakila monotherapy, kuma a cikin tsanani lokuta - tare da diuretics da sauran antihypertensive kwayoyi).
  • thyrotoxicosis (kawai wani bangare na hadaddun magani).
  • rigakafin angina harin da angina.
  • prophylaxis na migraine.
  • take hakkin cardiac kari (msl, arrhythmia, kuma paroxysmal supraventricular tachycardia, supraventricular tachycardia).
  • to rage hadarin mace-mace da kuma wajen kisa a cututtukan zuciya da kuma jijiyoyin zuciya jijiya cuta.
  • secondary rigakafin na tsokar zuciya infarction, kuma m tsokar zuciya infarction.
  • mitral bawul prolapse.
  • Dilated cardiomyopathy ne idiopathic.
  • zuciya da jijiyoyin jini giperkinez Essential, hyperkinetic cardiac ciwo, cuta na zuciya.

Reviews na medicament

Bisa ga sake dubawa na waɗanda suka taba kira da miyagun ƙwayoyi, da shi yadda ya kamata a magance da aiki da kyau sakamako a kan zuciya. Duk da haka, ya kamata a lura da cewa wasu marasa lafiya amsa magani ba sosai da kyau. Matsayin mai mulkin, wannan ne saboda da cewa shi yana da yawa contraindications da illa. Gaskiyar cewa a cikin marasa lafiya koka, bayyana a kasa a kan samu na kudi.

Contraindications da yin amfani da magani

Saboda haka, yanzu ka san abin da ake nufi da miyagun ƙwayoyi "Metoprolol" (alamomi ga yin amfani da aka bayyana kamar sama). Duk da haka, wannan magani yana da yawan contraindications. Wadannan sun hada da:

  • Mutum rashin ha} uri (Ina nufin hypersensitivity zuwa aiki ko karin aka gyara).
  • atrioventricular block 2nd da 3rd digiri.
  • daya-lokaci amfani da Mao hanawa.
  • kawancen sinuauricular.
  • bayyana Sistem sakulasan cuta (gefe).
  • sinus bradycardia (zuciya rate idan - akalla sittin da minti).
  • da qarancin ruwa da kuma labile nau'i na ciwon sukari.
  • rashin lafiya sinus ciwo.
  • haƙuri predisposed zuwa bronchospasm (Ina nufin, Bronchial fuka da kuma Bronchial wuce kima martani).
  • rayuwa acidosis.
  • hypotension (kasa da 100 mm Hg ..).
  • cardiogenic buga (da miyagun ƙwayoyi ba da shawarar ga marasa lafiya da ganewar asali "m tsokar zuciya infarction" ko da ake zargin shi).
  • m zuciya rashin cin nasara, na kullum (2nd da 3rd mataki) da kuma uncompensated.

Taƙaitawa akan yin amfani da miyagun ƙwayoyi (liyafar tare da matsananci hankali)

A abin da lokuta ya kamata a iyakance zuwa samun "Metoprolol" miyagun ƙwayoyi? Reviews masana sun ce wani kashi na medicament da za a rage a cikin hyperthyroidism, emphysema, rashin lafiyan tarihi, Bronchial fuka, wadanda ba rashin lafiyan mashako, psoriasis, pheochromocytoma, hanta cuta, koda da kuma (wani lokacin), ciki, myasthenia gravis da kuma janar maganin sa barci.

Shin yana yiwuwa a bayar da yara magani "Metoprolol"? A amfani da wannan magani da mutane a karkashin shekaru 18 da haihuwa da aka haramta. A ban a kan karbar kudi kara wa mata masu ciki da masu jego. Gaza bada hašin kai wadannan shawarwari, akwai wata babbar hadarin bradycardia, da qarancin ruwa da kuma hypotension a cikin jariri.

Idan kana bukatar wani kashi na magani a lokacin shayarwa, a cikin wannan lokaci na lactation ya kamata a katse.

Kwayoyi "Metoprolol" da "Metoprolol succinate": umarnin don amfani da

Yawanci, da medicament "metoprolol" kai a rana a cikin wani adadin 100 MG. A cikinsu ya ce girma ne zuwa kashi da dama allurai. A don cimma mafi kyau warkewa sakamako, da liyafar za a iya karu da sau 2. Duk da haka, matsakaicin kashi na miyagun ƙwayoyi kada wuce 400 MG.

Lokacin da daya-lokaci igiyar jini allura gudanar daga 2 zuwa 5 MG na cikin shirye-shiryen. A wannan yanayin, matsakaicin sashi ne 15-20 MG. A cikin rashi na so sakamako yarda ka sake-shigar da miyagun ƙwayoyi abu (a cikin minti 5).

Soke nadin da miyagun ƙwayoyi ya zama sauka a hankali. Yawanci wannan yana yi kwanaki goma a karkashin musamman dubawa na likita.

Harufan sashi daga cikin miyagun ƙwayoyi "metoprolol succinate" tare da supraventricular tachycardia, angina pectoris, arrythmia da hauhawar jini ne game da 50-100 MG sau daya a rana. Lokacin da goyon baya far da tsokar zuciya infarction samun medicament a kashi na 200 MG.

A m duration magani nufin "metoprolol succinate" ne watanni 3. Idan haƙuri ne kamu da kullum zuciya rashin cin nasara, da sashi ne gyara akayi daban-daban. Da farko, da miyagun ƙwayoyi ne a dauka a wani adadin 12.5 MG da zarar kullum don makonni 2, sa'an nan kuma kowane kwanaki 14, da kashi ne ninki biyu.

A gwada da kyau haƙuri a medicament ta matsakaicin ci a kowace rana zai iya isa 200 MG.

Side effects. shedu

Yana iya cutar da jiki magani "Metoprolol"? Reviews wannan shiri ya kunshi abubuwa da yawa na bayanai da cewa, bayan da m akwai mummunan sakamakon. Game da mamaki a tambaya?

  • Daga cikin juyayi tsarin: tsoka rauni, gajiya, yãyen mafarki, ciki, ciwon kai, tashin hankali, inda hakan na mota da hankulansu halayen, rage hankali, paresthesia a cikin extremities, gajere memory hanawa, drowsiness ko, conversely, rashin barci.
  • Daga cikin hankula: rage mugunya hawaye ruwa, rage hangen nesa, conjunctivitis, zafi da kuma bushe mucous membranes da idanu, ringing a cikin kunnuwa.
  • Cardio-jijiyoyin bugun gini tsarin: arrhythmia, sinus bradycardia, ƙarya angina, madugu disturbances infarction, ragewan jini, wata alama ce ta vasospasm, orthostatic hypotension, rage tsokar contractility da juwa.
  • Daga cikin tsarin narkewa kamar: bushe baki, ciki zafi, tashin zuciya, mahaukaci hanta aiki, maƙarƙashiya, amai, zawo, da kuma canje-canje a dandano.
  • Skin: itching, reversible alopecia, rash, flushing, rash, sweating, exacerbation na psoriasis, photodermatosis, exanthema da psoriasiform fata halayen.
  • Tsarin Numfashi: shortness na numfashi, hanci cunkoso, bronchospasm da wahala exhaling.
  • A wani ɓangare na da endocrine tsarin: hypothyroidism, da qarancin ruwa da kuma hyperglycemia.
  • Laboratory JARABAWA: thrombocytopenia, agranulocytosis, hyperbilirubinemia, leukopenia, kuma dagagge hanta enzymes.
  • A sakamako a kan tayin da mace mai ciki karkashin amfani: intrauterine girma retardation, bradycardia da qarancin ruwa da.

Bugu da kari, bayan samun ce miyagun ƙwayoyi wasu marasa lafiya bayar da rahoton abin da ya faru na hadin gwiwa zafi ko ciwon baya. Musamman rare show mutane cewa sun yi dan kadan ya karu jiki taro, rage libido ko iko.

Specific shiriya a kan yin amfani da miyagun ƙwayoyi

Yanzu a wani kantin magani za ka iya saya da miyagun ƙwayoyi "Metoprolol". A girke-girke da aka ba da ake bukata. Duk da haka, ga marasa lafiya shan magani ya kamata a kai a kai da sanya idanu kan malamin lafiyarka. Wannan shi ne musamman gaskiya ne ga waɗanda marasa lafiya da suke kamu da ciwon sukari ko angina.

An san cewa ta kara da sashi (fiye da 200 MG da rana) rage-rage cardioselective. A gaban zuciya rashin cin nasara far an fara kawai bayan da diyya mataki ne kai.

Mutanen da suka yi amfani da lambar sadarwa ruwan tabarau, dole ne ka yi la'akari da cewa a cikin mahallin da magani, "metoprolol" rage samar da lachrymal ruwa.

Wani lokaci wannan magani masks wasu cututtuka na hyperthyroidism. A wannan zato karbo daga cikin miyagun ƙwayoyi a marasa lafiya tare da ya ce cutar da aka contraindicated, tun da shi kara habaka da cututtuka.

Idan ya cancanta, da aiki da haƙuri kamata ko da yaushe faɗakar da anesthesiologist miyagun kwayoyi far.

A lokacin jiyya, da wani magani, "metoprolol" wajibi ne a ci dace tufafi. Wannan shi ne saboda cewa da miyagun ƙwayoyi iya haifar da rashin lafiyan halayen ga fata saboda daukan hotuna zuwa ga hasken rana.

Ba za mu iya ce cewa magani "Metoprolol" (analogues wannan magani musamman) a cikin tsofaffi zai iya sa bayyanar da kara bradycardia, alama raguwa a jini, atrioventricular block. Wannan shi ne dalilin da ya sa wadannan marasa lafiya na bukatar musamman iko.

Bugu da kari, a lokacin jiyya da wannan magani ya kamata dena tuki wani abin hawa da kuma dakatar azuzuwan m ayyuka da cewa bukatar babban taro da psychomotor gudun halayen. Haka kuma an bada shawarar cewa m na ethanol.

Data kasance miyagun ƙwayoyi analogs

Abin da idan haƙuri shi ne iya sayan magani wajabta ta likita, "metoprolol"? Its analogues suna samuwa a wani kantin magani. Mafi yawansu ba su dauke da wani irin aiki abu, haka shi yana da guda Properties kamar yadda ya ce miyagun ƙwayoyi. Daga cikin wadannan za a iya ambata da wadannan kwayoyi: "Metoprolol Acre", "Metolol", "Metokor Adifarm" da sauransu.

Bayan data saye nufin wani haƙuri rika koma zuwa a haɗe umarnin, kuma domin ganawa da wani likita. Wannan shi ne saboda cewa da samun nufin iya bambanta daga sama dosages wajen.

Abin da kuma ya aikata da wannan magani analogs? Sauya likita ta nada nufin iya zama da wadannan magunguna: "bisoprolol" "Metoprolol-ratiopharm", "Metokard", "Korvitol", "Metozok", "Lidalok", "Serdol", "Egilok", "Emzok" da sauransu.

Yadda za a adana da kuma nawa magani?

Yanzu da ka san abin da ake nufi, da yadda kuma a cikin abin da sashi dauki magani "Metoprolol". Adana shi a wani sanyi wuri (msl, a wani firiji) ko wani dakin inda zafin jiki ba ya wuce 25 digiri. A wannan yanayin, da miyagun ƙwayoyi ya kamata a kiyaye shi daga hasken rana kai tsaye.

Shiryayye rayuwar ce miyagun ƙwayoyi da kuma mafiya yawa daga ta takwarorinsu na shekaru biyar daga ranar samar. Bayan wannan lokaci, da magani amfani da warkewa da kuma prophylactic dalilai da aka haramta. Ya kamata a jefar.

Similar articles

 

 

 

 

Trending Now

 

 

 

 

Newest

Copyright © 2018 ha.atomiyme.com. Theme powered by WordPress.