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"Bisoprolol-Prana": alamomi don amfani, analogs, reviews, umarnin don amfani. "Bisoprolol-Prana" da "bisoprolol": sabanin

Akwai da yawa magunguna a kan tushen da bisoprolol, wanda aka samu nasarar yi amfani da magani na cutar hawan jini da kuma gazawar da zuciya tsoka. Daga cikinsu akwai m samfurin "bisoprolol-Prana".

fasalin

Samar da zabe beta adrenoblokatornoe nufi da Rasha kamfanin OOO "PRANAFARM".

An samar a cikin nau'i na zagaye, biconvex Allunan cewa da rabuwa shafi da kuma wani fim shafi.

A lokacin da ka yi amfani da "bisoprolol-Prana" umarnin don amfani - Wannan shi ne abu na farko da za ka bukatar kula. A miyagun ƙwayoyi ne samuwa a cikin wadannan dosages: 5 da 10 MG. Launi Shell karami Allunan kodadde rawaya, da kuma manyan - kodadde orange. Da abinda ke ciki na miyagun ƙwayoyi ne kusan fararen.

tsarin

Daya kwamfutar hannu miyagun ƙwayoyi "bisoprolol-Praana" kamar yadda mukaddashin abu dauke 5 da 10 MG bisoprolol hemifumarate. A gaban magnesium stearate, masara sitaci, microcrystalline cellulose tsarin, Crospovidone, colloidal silicon oxide, alli phosphate dehydrated form damar da medicament da kuma samar da muhimman solubility da bioavailability.

A fim mai rufi sashi na 5 MG na baƙin ƙarfe oxide ba rawaya, polyethylene glycol (sa 400), titanium dioxide, silicone. A shafi wanda ƙunsa da kwaya manyan, akwai wani colorant a cikin nau'i na ja da baƙin ƙarfe oxide.

inji na mataki

By zabe beta adrenoblokatornym nufin cewa ba su da nasu sympathomimetic aiki irin, sun hada da "bisoprolol-Prana". Umurnai na amfani bayyana ta pharmacodynamic halaye. Allunan da wani sakamako a kan rage matsin lamba, daidaita da kari kuma kawar da tsoka ischemia. Lokacin da kulle a cikin kananan dosages zuciya tsoka mai amsa sigina beta miyagun ƙwayoyi adrenozavisimyh 1 ne a rage samar da cyclic adenosine monophosphate da alli ions a cikin cell halin yanzu. Har ila yau, wani karu a zuciya kudi da kuma rage ta mita, damuarn da matakai hade da watsin da excitability.

Hypotensive effects nuna a ma low da darajar da cewa ma'anar da minti girma jini wurare dabam dabam, rage tasiri a kan gefe jijiyoyin bugun gini gado. Rage high matsa lamba auku bayan 'yan kwanaki, kamar yadda ya cancanta don daidaita biyu-wata jiyya matakai.

Antiarrhythmic effects bayyana a kawar da dalilai da cewa karya da bugun zuciya. Wadannan sun hada da jihar tachycardia, waye aiki na m juyayi tsarin a sashen, ta ƙara matakan cyclic adenosine monophosphate, jijiya hauhawar jini.

alamomi

Kafin yin amfani da shi wajibi ne, don su bincika, domin wanda kungiyoyin na marasa lafiya ne "bisoprolol-Prana". Alamomi Associated da antianginal sakamako. Shi ne saboda kasa bukatar cardiac tsokar oxygen kwayoyin ta rage ƙanƙancewa mita, ta ƙara jini ya kwarara da kuma lokaci a diastole.

Mene ne sakamakon wannan miyagun ƙwayoyi a matsayin kwaya "bisoprolol-Prana", daga abin da suke yi? Ganin pharmacological halaye, su ana amfani da:

  • lura da hauhawar jini.
  • ischemic cututtukan zuciya.
  • angina a irin ƙarfin lantarki.
  • Sakandare rigakafin na tsokar zuciya infarction:
  • gazawar da kullum irin.

Ga sasannin wanda shi ne kyawawa don amfani "bisoprolol-Praana" miyagun ƙwayoyi. Alamu suna hade da illa cardiac yi. Wadannan sun hada da wani karuwa a sinus kari, supraventricular da kuma na ramin zuciya arrhythmias, canza zuciya tare da mitral bawul protrusion irin da hyperthyroidism.

A takamaiman amfani da miyagun ƙwayoyi

Umarnin don amfani "bisoprolol-Prana" ya bada shawarar da magani da safe kafin karin kumallo, da dukan ba tare da daukan taban.

Domin lura da hauhawar jini, cardiac ischemia da kuma hana wani yanayin angina amfani guda kashi a kashi kwamfutar hannu hada da 5 MG bisoprolol. Idan ya cancanta, da sashi ne ninki biyu, amma kuma za a iya amfani da shi kadai. Max bisoprolol kada wuce 20 MG kullum kullum.

Kawai wani likita zai iya rubũta sashi da kuma liyafar nufin "bisoprolol-Prana". Alamomi dole a bi umarnin da miyagun ƙwayoyi. Kafin nada rajistan shiga mita na contractions daga cikin zuciya tsoka. Ability don daidaita yawan Allunan bayan nazarin warkewa martani.

Mutane da yawa marasa lafiya mamaki game da ko yana yiwuwa "bisoprolol-Prana" bisect. A gaban da SEPARATOR ba da wata dama don rage kwaya idan kana bukatar wani daban-daban sashi.

Don kawar kullum zuciya maye irin makon farko ta amfani 1.25 MG bisoprolol. Irin wannan kashi za a iya samu ta hanyar rarraba da Allunan, dauke da 2.5 MG na aiki abu. Duk da haka, shi yana zuwa fara far da sauran manufacturer, a matsayin wata hanya ta "Bisoprolol-Praana" da aka bayar kawai 5 da 10 MG. A lokacin da na biyu mako gudanar 2.5 MG. Tare da kwanaki 14 na lura da shan 3,75 MG na miyagun ƙwayoyi. A karo na hudu mako da sashi aka ƙara zuwa 5 MG, da kuma bayan watanni biyu na far amfani da 7.5 MG bisoprolol. Goma sha biyu mako fara da kashi na 10 MG.

Idan haƙuri yana da daban-daban tafka magudi a koda ko hanta, da kuma dabi'u na creatinine yarda kasa da 20 ml for 1 minti daya, sa'an nan matsakaicin za a iya gudanar up to 10 MG da miyagun ƙwayoyi.

A lokacin shirya aiki bisoprolol soke na kwana biyu, don haka shi ba zai shafi maganin sa barci. Idan kwamfutar hannu ya kasance bugu, da zabi irin wakili don zafi, wanda farfado inotropic effects, korau m adadin.

Lokacin da wani tsofaffi haƙuri akwai wani hari bradycardia da zuciya rate kasa da 52 lashe minti daya, jijiya hypotension da systolic matsa lamba kasa da 100 mmHg, bronchospasm, na ramin zuciya arrhythmia, illa hanta da na koda aiki, to, bãbu wani karu sashi har jimlar an daina. bisoprolol togiya iya haifar da ci gaban mai depressive jihar, wanda aka sa ta data daga cikin beta-shafi.

Mazan mutane bã su ciyar da wata sashi gyara.

Ka guji zato katsewa na magani, wanda zai iya sa da ci gaban mai tsanani arrhythmias ko tsokar zuciya infarction yanayin tsokoki. Kau da miyagun ƙwayoyi ne da za'ayi da hankali rage da kashi for 14 days. Kwanaki uku iya rage sashi daga 25%.

Features na magani

Don amfani da "bisoprolol-Prana" wa'azi a kan aikace-aikace hada da jerin matakan da cewa sarrafa jihar na rashin lafiya mutum. Wadannan sun hada da kullum a cikin matakin farko na definition na zuciya kudi da kuma jini ji, to, wanda aka bari bayan watanni uku. Sauran muhimmanci Manuniya ne electrocardiogram da jini sugar matakan da masu ciwon sukari, wanda mataki ba fiye da 5 months.

Mazan marasa lafiya bukatar lokaci-lokaci monitoring da kodan, wanda yana da za'ayi bayan 4 watanni.

Jiyya na kullum zuciya maye a cikin na farko mataki na karbar low kashi na bukatar wani hudu-hour jarrabawa na haƙuri, cikinsa da mita da aka bari by tsokar ƙanƙancewa, jini ko electrocardiograms.

Kafin nada magani da bisoprolol haƙuri sanar da yadda za a lissafta da zuciya rate. A cikin hali na low dabi'u na index (har zuwa 50 lashe da minti) da ake bukata shawarar likita.

Har ila yau, a kwatanta mataki "bisoprolol-Prana" miyagun ƙwayoyi jagora ya hada da bayani a kan bukatar nazarin cewa sanin da waje numfashi ga marasa lafiya da bronchopulmonary cututtuka.

Ba dukan marasa lafiya da beta-adrenoblokatornye kwayoyi taimaka bi angina. Saboda su gazawar gaban tsanani jijiyoyin zuciya atherosclerosis, ischemic ciwon low bakin kofa. A wannan yanayin, da zuciya rate ne kasa da 100 lashe minti daya, da kuma a can ne da karuwa a karshen-diastolic girma na hagu ventricle tare da take hakkin subendocardial jini ya kwarara. Smoking mutane bisoprolol kuma taimaka muni.

Mutane da bronchospastic cuta, irin cardioselective wajabta wajen, idan akwai rashin ha} uri ga low dace da kuma kwayoyi da rage matsin lamba. A hali na yawan abin sama akwai wani babban Yiwuwar Bronchial spasm.

Lokacin zalunta marasa lafiya da thyrotoxicosis beta-shafi, da yiwuwar masking mutum na asibiti ãyõyin wuce kima thyroid aiki, musamman tachycardia. Irin wannan marasa lafiya ba zai iya zana kaifi soke wani shiri, domin ya hana karawa da cututtuka.

Idan marasa lafiya saka lambar sadarwa ruwan tabarau, da liyafar na bisoprolol zai iya sa wani karu a samar da hawaye ruwa, wanda na bukatar karin musamman ido saukad instillation.

Lokacin da miyagun ƙwayoyi da ake amfani, marasa lafiya da pheochromocytoma, ƙila a sami wata paradoxical hauhawar jini. A irin wannan yanayi da na farko alpha adrenoblokadnoe mataki.

A gaban ciwon sukari masks bouts na tachycardia ya sa wani karu a matakin glucose a cikin jini jini. Da yake zabe beta-shafi, da miyagun ƙwayoyi ne ba iya bunkasa insulin hypoglycemic yanayin da impede da daidaita da glucose matakin da ake so dabi'u.

Catecholamines, normetanephrine, antinuclear antibodies da vanillylmandelic acid a cikin jini da kuma fitsari da aka ƙayyade ne kawai a wariya nufin "bisoprolol-Praana".

Ga ciki kuma lactating mata, da nada da miyagun ƙwayoyi da aka za'ayi shan la'akari da amfanin da masu juna biyu kwayoyin, amma akwai yiwuwar illa a cikin tayi.

Wannan magani an contraindicated?

Allunan "bisoprolol-Prana 'umarnin don amfani ba rika amfani da ƙara laulayi, m ko na kullum decompensated insufficiency na zuciya tsoka, bugu cardiogenic, kawancen sinuauricular da atrioventricular biyu da na uku irin, a wani ciwo hade da rauni a cikin sinus kumburi, m bugun zuciya tare da wani tsanani kasa da 60 lashe.

Contraindication ne gaban:

  • cardiomegaly tare da kara girman da kuma nauyi na zuciya tsoka.
  • rage matsa lamba a cikin jijiyoyi da wani systolic darajar kasa da 90 mm Hg.
  • kullum obstructive na huhu cuta.
  • Bronchial fuka.
  • cuta jini wurare dabam dabam a gefe tasoshin a baya, saukarwa.

wašanda ba'aso sequela

Medicine "bisoprolol-Praana" zai iya sa daban-daban gefen sakamakon abin da ta shafi tsakiyar yankin da kuma na gefe m tsarin. Sun bayyana ciwon kai, gajiya, barci tsangwama gwamnatin, tawayar yanayi da kuma hallucinations.

A ke so matakai a cikin zuciya da jini saboda da orthostatic hypotension, flushing, sweating, palpitations jinkiri da kuma rashin tsokar aiki.

Sauran manifestations illa ne don rage mugunya na lacrimal gland, conjunctivitis ci gaba, zawo, itching na fata, maƙarƙashiya, tashin zuciya, tsoka rauni da cramps. Obstructive cututtuka na iya faruwa a cikin bronchi.

kama preparty

Original kayan aiki a kan tushen da bisoprolol ne Allunan "Concor". Suna samar da Jamusanci kamfanin "Merck".

Bisa ga wannan miyagun ƙwayoyi da aka ɓullo da irin wannan shirye-shirye, dauke da matsayin aiki abu bangaren bisoprolol fumarate.

Rasha miyagun ƙwayoyi masana'antun sarrafa beta-blockers tare da daban-daban cinikayya sunayen. An misali zai zama a wajen "Bisoprolol-Praana": da analogs da sashi na 2.5 MG, 5 MG da 10 MG. Wadannan kwayoyi hada da Allunan:

  • "Bisogamma".
  • "Niperten".
  • "Kordinorm".
  • "Biprol".

Wadannan kayan aikin an kuma samar da kamfanonin ketare. A pharmaceutical kasuwar buga kayayyakin, da lakabi na wanda yanzu sunan sha'anin, misali, "bisoprolol-Teva", "bisoprolol-Ratiopharm," "bisoprolol-Sandoz", "bisoprolol-warai."

Akwai analogues, wanda ake kira kawai "bisoprolol". Irin wannan magunguna kerarre da Rasha shuke-shuke: JSC "kokuwa", JSC "Arewa Star", LLC "lemar sararin samaniya Pharmaceuticals", JSC "Biocom".

Idan muka kwatanta da kwaya "bisoprolol" da "bisoprolol-Prana", bambanci zai kasance a cikin ingantaccen da kuma gwada yawa abun da ke ciki karin aka gyara. Irin bambance-bambance ba zai shafi permeability da bioavailability na aiki dũkiyõyinsu a cikin jiki, ya kuma inganta, da warkewa sakamako daga cikin miyagun ƙwayoyi zai zama guda.

reviews

Mutane da yawa marasa lafiya lura saukaka amfani da magunguna dauke da bisoprolol, saboda sun kawai dauki sau daya a rana. Daya kwamfutar hannu isa ga wani yini guda domin daidaita jini.

Game da nufin "bisoprolol-Prana" mai kyau sake dubawa. Su ne shaida ta high selectivity, wanda shi ne dalilin da ya sa kwayoyi yana tare da m illa idan aka kwatanta da sauran beta-blockers.

Marasa lafiya lura amfani da rare illa da taimakawa ga gwamnatin rikon kwarya a wasu marasa lafiya neman magani bisa ga miyagun ƙwayoyi.

Maza ce cewa da miyagun ƙwayoyi ba sa disturbances na iko. Bugu da kari, wannan al'amari an tabbatar ta hanyar yawa karatu.

Drug "bisoprolol-Prana" ya nuna na rayuwa saka hannu a game da cholesterol, triglyceride kuma glucose metabolism. Wannan dukiyar yale mu mu rubũta ta ga marasa lafiya da na biyu da irin ciwon sukari ko wani predisposition zuwa ƙãra glucose matakai a cikin jini. Haka kuma, irin wannan marasa lafiya kuma bar tabbatacce feedback game da miyagun ƙwayoyi.

Saboda da kananan yawan m halayen kwayoyi wajabta ga marasa lafiya a cikin tsofaffi. Marasa lafiya suna da'awar cewa da miyagun ƙwayoyi inganci da kuma aminci daga sauran antihypertensives Beta blokatornogo jerin.

A amfani da miyagun ƙwayoyi "bisoprolol-Prana" ne da low price, wanda shi ne samuwa ga low-samun kudin shiga mutane, wanda kuma ya nuna a cikin m martani.

Amma duk da dukan abũbuwan amfãni daga Allunan, kawai likita Can rubũta su dangane da binciken sakamakon.

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