Kiwon lafiyaShirye-shirye

Product "Levodopa": umarnin don amfani, description, abun da ke ciki, analogs da kuma sake dubawa

Mene ne magani "Levodopa"? Umarnin don amfani, price, reviews game da miyagun ƙwayoyi za a tattauna kadan kara. Za ka kuma koyi game da abin da aka wajabta wannan magani, idan ya na da wani m halayen da kuma contraindications, a cikin abin da ya samar da shi ne don sayarwa, wanda aka hada da a cikin abun da ke ciki, da sauransu.

A abun da ke ciki, siffar, description

Wanne aka gyara ƙunshi wani magani "Levodopa"? Umurnai na amfani nuna cewa aiki sashi daga cikin miyagun ƙwayoyi ne levodopa. A sale shi ne a cikin nau'i na madauwari spigot Allunan farin launi, kunsasshen a kwane-kwane cell da kwali kwalaye, bi da bi.

Ka'idar aiki na wani medicament

miyagun ƙwayoyi "Levodopa" Yaya ta yi aiki? Umarnin don amfani, reviews sun ruwaito cewa wannan hade antiparkinsonian wakili. Yana da nufin kawar da rigidity, hypokinesia, tremor, drooling da dysphagia.

A cikin jiki, mukaddashin magani bangaren da aka tuba zuwa dopamine (CNS), game da shi sa up karancin kashi.

Dopamine da ya auku a gefe kyallen takarda, ya nuna babu anti-Parkinson effects na levodopa. Wannan shi ne saboda da cewa shi ba ya shiga cikin tsakiyar m tsarin da yake da manyan dalilin m halayen da miyagun ƙwayoyi.

Don rage kashi na aiki abu a jikin mutum da ake sa medicament a hade tare da mai hanawa na gefe dopa-decarboxylase. Wannan dabara taimaka wajen rage illa daga shan kwayoyi.

Pharmacokinetics

Nawa magani da ake tunawa "Levodopa"? Umarnin a kan aikace-aikace jihohin da bayan samun da miyagun ƙwayoyi a cikin jikin shi aka quite hanzari tunawa daga hanji.

Absorption na aiki abu ne game da 20-30%. A wannan warkewa sakamako da aka lura bayan game 3 h.

Abinci ci (ciki har da wani abinci) kai tsaye rinjayar da sha da miyagun ƙwayoyi.

Da miyagun ƙwayoyi ne metabolized, game da shi, kafa da dama metabolites. Tukar tumbi da aiki abu faruwa ta hanyar da kodan, kuma ta hanyar da hanji.

alamomi

A karkashin abin da yanayi marasa lafiya wajabta da miyagun ƙwayoyi "Levodopa"? Umurnai na amfani bisa ga wadannan alamomi:

  • postencephalitic ciwo da ya auku a cerebrovascular cututtuka ko mai guba maye.
  • Parkinson ta ciwo, haka ma, wanda aka sa ta yin amfani da antipsychotic kwayoyi.
  • Parkinson ta cutar.

contraindications

Ko akwai contraindications a "L-dopa" miyagun ƙwayoyi? Umarnin don amfani da rahoton cewa wannan magani an haramta kai a cikin wadannan lokuta:

  • hypersensitivity da aka gyara.
  • a hade tare da Mao hanawa.
  • a lokacin daukar ciki da kuma a lokacin da nono-ciyar da wata baby.
  • marasa lafiya karkashin shekaru 18.

Tare da babban kula da miyagun ƙwayoyi za a iya nada a:

  • emphysema.
  • gaban cutar huhu, cututtukan zuciya, hanta da kuma tsarin endocrine da receptacles.
  • Bronchial fuka.
  • bayyananen na psychosis.
  • melanoma (ciki har da tarihi).
  • kwana-ƙulli glaucoma.
  • maimaita seizures (convulsions).
  • bude-kwana glaucoma, wanda ya auku a kullum form.
  • koda da hanta gazawar;
  • tsokar zuciya infarction (tarihi), da kuma a cikin siffofin daban-daban iri arrhythmias.
  • duodenal miki da ciki;
  • CNS manifestations na zalunci;
  • zuciya kari disturbances.

A miyagun ƙwayoyi ne "L-dopa": umarnin don amfani da

Description da miyagun ƙwayoyi da aka gabatar a sama. Kamar yadda ya kamata?

Bisa ga umarnin, da miyagun ƙwayoyi ne riƙi baki. A sashi ne a hankali ya karu daga m zuwa matsakaicin (dangane da mutum haƙuri).

Fara lura da wani kashi na 0.25-1 g Wannan adadin ne zuwa kashi uku rabo. A sashi ne a hankali ya karu zuwa 0,125-0,75 g Shin, shi a daidai lokaci na lokaci (msl, kwanaki uku), mayar da hankali a kan mutum haƙuri ta mayar da martani, har zuwa lokacin da ya a lokacin da ganiya sakamako za a lura daga far.

A kalla kashi da rana kada wuce takwas grams.

Magani a wani hali, kada soke gunaguni ƙwarai. Tsaya shan shi a hankali.

m halayen

Shin da gefen sakamakon da miyagun ƙwayoyi "Levodopa"? Umurnai na Amfani furta cewa, a cikin mahallin da liyafar a mutum na iya fuskanci wasu m halayen da rinjayen aiki na duk tsarin na jiki:

  • Zuciya da jijiyoyin jini tsarin: zuciya palpitations, arrhythmia, tashin hankali na matsa lamba, orthostatic halayen, syncope, da sauransu.
  • Narkewa kamar fili: zawo da amai, dyspepsia, anorexia, maƙarƙashiya, canji a dandano, bushe baki, zubar da jini daga cikin gastrointestinal fili.

Ya kamata kuma a lura da cewa ba cire gefen halayen shafi aiki na hematopoiesis, urinary, na numfashi, da kuma juyayi tsarin. Sau da yawa a cikin marasa lafiya da samun wannan magani rashin lafiyan halayen faruwa, canji a dakin gwaje-gwaje sigogi da makaruhai effects a kan fata.

Lokuta da yawan abin sama (bayyanar cututtuka, magani)

A da ake ji high allurai nuna wani gagarumin kayan haɓɓaka aiki na gefe effects. Irin wannan yanayi bukatar magani a cikin wani nau'i na lavage, haƙuri da janar yanayin da lura da kuma aiki da zuciya. Idan ya cancanta, gudanar da wani antiarrhythmic far.

miyagun ƙwayoyi interactions

Lokaci daya liyafar da kuma la'akari da shirye-shiryen "ditilina" beta-agonists, da kuma jamiái cewa an yi nufi ga inhalation maganin sa barci, qara da alama na arrhythmias na zuciya.

Bioavailability "Levodopa" na iya rage tricyclic antidepressants.

A hade da miyagun ƙwayoyi da "thioxanthenes," "Diazepam" antipsychotic "Phenytoin" m-holinoblokatorami "clonidine", "Difenilbutilpiperidinom" "Papaverine", "Clozapine", "phenothiazine" "pyridoxine" da "reserpine" quite sau da yawa shi na rage antiparkinsonian sakamako.

Lithium formulations kara yiwuwar faru na dyskinesias da hallucinations, da kuma "methyldopa" medicament qara gefen halayen.

A hade da Mao hanawa da kuma "Levodopa" kaiwa zuwa illa wurare dabam dabam. A wannan batun, da tazara tsakanin allurai da wadannan magunguna dole ne a kalla 14 days.

Alama raguwa a matsa lamba ta lura da wani hade da magani dauke "tubocurarine".

Drug "metoclopramide" kara bioavailability "Levodopa" accelerating ciki emptying. Wannan na iya adversely shafi cikin shakka daga cikin cutar.

Specific shawarwari don amfani da miyagun ƙwayoyi

Me kana bukatar ka sani kafin shan da Allunan, "Levodopa"? Umurnai na amfani (da farashin kasa) yayi kashedin game da barazana ga lafiya da na ba zato soke wata medicament.

A lokuta inda ba shi yiwuwa su kauce wa rage daga cikin sashi ko karbo daga magani bukatar yau da kullum saka idanu na haƙuri da yanayin.

Kafin da miyagun ƙwayoyi ba da shawarar zuwa cinye abinci mai arziki a cikin furotin, tun da shi ya rage absorbability na aiki abu.

A far bukatar ci gaba da sa ido na daban-daban tsarin, gabobin, da kuma jini sigogi.

Price da analogues

A mafi kusa analogues "L-dopa" shiri na nufin shi ne kamar wani "levodopa benserazide" da "Levodopa Carbidopa". Umarnin don amfani da rahoton cewa wadannan kwayoyi da wannan alamomi, illa, sunadaran da mataki da contraindications. Iyakar abin da bambanci tsakanin wadannan kudi ne abun da ke ciki.

Irin wannan aiki abubuwa kamar carbidopa da benserazide rage samar da dopamine a gefe nama, game da shi kara yawan levodopa shigar da CNS.

Saboda haka, zai iya a amince a lura da cewa prescriptions "Levodopa Carbidopa" da "levodopa benserazide" (umarnin don yin amfani da wadannan hanyoyi suna kuma saka a cikin marufi) gusar ƙarin liyafar hanawa gefe dopa-decarboxylase.

Amma ga sauran takwarorinsu, sa'an nan da karshen hada da irin kwayoyi a matsayin "Isik Meath", "Tremonorm", "Dopar 275", "Tidomet", "Duellin ',' Sinemet ',' Zimoks", "Sindopa", "Isik" "Lac". Dole ne su sanya kawai likita.

Farashin "Levodopa" da miyagun ƙwayoyi ne quite high. A Pharmacy, za ka iya saya da wannan magani a cikin 1500-1850 rubles.

magani Reviews

Jiyya na wani cuta ya kamata a za'ayi ne kawai don dalili na wani gogaggen likita. Kuma Parkinson ne ba togiya.

Marasa lafiya da suke dauki da miyagun ƙwayoyi "Levodopa" a cikin tafin kafa hankali, kuma ba su da wani m warkewa sakamako. Saboda haka sau da yawa wannan medicament sake dubawa ne korau. Masu amfani sun ruwaito cewa ko da tare da shafe tsawon amfani da magunguna sananne inganta sun kyau kiyaye.

Idan magani ake dauka a karkashin shawara da makirci, wanda aka ci gaba da wani gogaggen sana'a ne wadannan da hanya da cuta, da jiyya tsari ne kusan ko da yaushe nasara. Wannan shi ne saboda cewa da aiki miyagun ƙwayoyi ne a dauka a cikin wani m sashi, wanda ya dogara a kan haƙuri, da halaye da cutar da kuma wasu dalilai.

Marasa lafiya suna tsananin kaucewa lura regimen, sun ruwaito cewa miyagun ƙwayoyi "Levodopa" ne sosai tasiri a kawar da matsalar lafiya.

A gaskiya, da yawa koka game da tsadar kudin magani. Duk da haka, masana da'awar cewa farashin wannan miyagun ƙwayoyi ne gaba daya wajaba a kansa.

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